A Diels-alder Route Towards Pyrimidin-4-ones

Bayard, Philippe;Sainte, Francy;Beaudegnies, R.;Ghosez, Léon
(1988) Tetrahedron Letters — Vol. 29, n° 31, p. 3799-3802 (1988)

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Authors
  • Bayard, PhilippeUCLouvain
    Author
  • Sainte, FrancyUCLouvain
    Author
  • Beaudegnies, R.UCLouvain
    Author
  • Ghosez, LéonUCLouvain
    Author
Abstract
N-acylimidates are readily silylated with t-butyldimethylsilyl triflate in the presence of triethylamine to give 2-aza-1,3-dienes. These react with activated nitriles to yield pyrimidin-4-ones.
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Bayard, P., Sainte, F., Beaudegnies, R., & Ghosez, L. (1988). A Diels-alder Route Towards Pyrimidin-4-ones. Tetrahedron Letters, 29(31), 3799-3802. https://doi.org/10.1016/S0040-4039(00)82118-8 (Original work published 1988)