Asymmetric Amination of Carboxylic-acids Via a Diels-alder Strategy

Gouverneur, Véronique;Ghosez, Léon
(1991) Tetrahedron Letters — Vol. 32, n° 39, p. 5349-5352 (1991)

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  • Gouverneur, VéroniqueUCLouvain
    Author
  • Ghosez, LéonUCLouvain
    Author
Abstract
2-azadienes 1 which are readily prepared from acyl chlorides react with high facial selectivity with the chiral carbamoyl nitroso dicnophile 2. Reduction and hydrolysis of the adducts yield enantiomerically pure amino acids.
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Gouverneur, V., & Ghosez, L. (1991). Asymmetric Amination of Carboxylic-acids Via a Diels-alder Strategy. Tetrahedron Letters, 32(39), 5349-5352. https://doi.org/10.1016/S0040-4039(00)92382-7 (Original work published 1991)