Green synthesis of benzamides in solvent- and activation-free conditions

Alalla, A.;Merabet-Khelassi, M.;Aribi-Zouioueche, L.;Riant, Olivier
(2014) Synthetic Communications : an international journal for rapid communication of synthetic organic chemistry — Vol. 44, n° 16, p. 2364-2376 (2014)

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Authors
  • Alalla, A.
    Author
  • Merabet-Khelassi, M.
    Author
  • Aribi-Zouioueche, L.
    Author
  • Riant, OlivierUCLouvain
    Author
Abstract
Herein, we describe a clean and ecocompatible pathway for both N-benzoylation and N-acetylation of anilines, amines, diamines, and aminoalcohols using three enol esters with good yields. We have improved the use of vinyl benzoate for the direct introduction of a benzamido-moiety under solvent- and activation-free conditions. The recovered amides are easily isolated by crystallization. Copyright © 2014 Taylor & Francis Group, LLC.
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Alalla, A., Merabet-Khelassi, M., Aribi-Zouioueche, L., & Riant, O. (2014). Green synthesis of benzamides in solvent- and activation-free conditions. Synthetic Communications : an international journal for rapid communication of synthetic organic chemistry, 44(16), 2364-2376. https://doi.org/10.1080/00397911.2014.898072 (Original work published 2014)